Terfenadine

CAS No. 50679-08-8

Terfenadine ( MDL 9918; NSC 665802; (±)-Terfenadine; DL-Terfenadine )

Catalog No. M14729 CAS No. 50679-08-8

Terfenadine is a histamine H1-receptor antagonist, which blocks HERG and KATP (KIR6) channels.

Purity : >98%(HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
50MG 32 In Stock
100MG 45 In Stock
200MG 68 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Terfenadine
  • Note
    Research use only, not for human use.
  • Brief Description
    Terfenadine is a histamine H1-receptor antagonist, which blocks HERG and KATP (KIR6) channels.
  • Description
    Terfenadine is a histamine H1-receptor antagonist, which blocks HERG and KATP (KIR6) channels.
  • Synonyms
    MDL 9918; NSC 665802; (±)-Terfenadine; DL-Terfenadine
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    HT; mAChR; Potassium Channel
  • Research Area
    Inflammation/Immunology
  • Indication
    ——

Chemical Information

  • CAS Number
    50679-08-8
  • Formula Weight
    471.67
  • Molecular Formula
    C32H41NO2
  • Purity
    >98%(HPLC)
  • Solubility
    Water: 0.0963 mg/L
  • SMILES
    OC(C1=CC=C(C(C)(C)C)C=C1)CCCN2CCC(C(C3=CC=CC=C3)(O)C4=CC=CC=C4)CC2
  • Chemical Name
    1-(4-(tert-butyl)phenyl)-4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)butan-1-ol

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Kishimoto W, et al. Res Commun Mol Pathol Pharmacol. 1997 Dec;98(3):273-92.
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