Tecastemizole

CAS No. 75970-99-9

Tecastemizole ( Norastemizole; R 43512; R-43512; R43512; T 1348 )

Catalog No. M27833 CAS No. 75970-99-9

Tecastemizole is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 192 Get Quote
10MG 282 Get Quote
25MG 480 Get Quote
50MG 691 Get Quote
100MG 972 Get Quote
500MG 1944 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Tecastemizole
  • Note
    Research use only, not for human use.
  • Brief Description
    Tecastemizole is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.
  • Description
    Tecastemizole is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.
  • Synonyms
    Norastemizole; R 43512; R-43512; R43512; T 1348
  • Pathway
    GPCR/G Protein
  • Target
    Histamine Receptor
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    75970-99-9
  • Formula Weight
    324.4
  • Molecular Formula
    C19H21FN4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Fc1ccc(Cn2c(NC3CCNCC3)nc3ccccc23)cc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Bernd R?dle, et al.Metabolic labeling of newly transcribed RNA for high resolution gene expression profiling of RNA synthesis, processing and decay in cell culture. J Vis Exp. 2013 Aug 8;(78):50195.
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