Talinolol( (±)-Talinolol )

Catalog No. M27440 CAS No. 57460-41-0

(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.

Purity : >98% (HPLC)

COA

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HNMR

HPLC

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Biological Information

Product Name

Talinolol
Note

Research use only, not for human use.
Brief Description

(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
Description

(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
In Vitro

Human OATP1A2-, rat Oatp1a5-, and rat Mdr1a-mediated Talinolol transport can be inhibited by naringin, with IC50s of 343, 12.7, and 604 μM, respectively, in LLC-PK1 cell and Xenopus laevis oocyte systems.
In Vivo

Talinolol (20 mg/kg; i.p.) plasma and liver AUC0-5 h are increased by Zosuquidar administration.Bioavailability of Talinolol can be enhanced by coadministration with grapefruit juice (GFJ) in rats.
Synonyms

(±)-Talinolol
Pathway

Angiogenesis
Target

Adrenergic Receptor
Recptor

——
Research Area

——
Indication

——

Chemical Information

CAS Number

57460-41-0
Formula Weight

363.502
Molecular Formula

C20H33N3O3
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 100 mg/mL (275.11 mM)
SMILES

CC(C)(C)NCC(O)COc1ccc(NC(=O)NC2CCCCC2)cc1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Asano T, Murayama T, Hirai Y, Shoji J. Comparative studies on the constituents of ophiopogonis tuber and its congeners. VIII. Studies on the glycosides of the subterranean part of Ophiopogon japonicus Ker-Gawler cv. Nanus. Chem Pharm Bull (Tokyo). 1993;41

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