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TRPM4-IN-1

CAS No. 351424-20-9

TRPM4-IN-1( CBA | 4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid )

Catalog No. M24301 CAS No. 351424-20-9

TRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    TRPM4-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    TRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.
  • Description
    TRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.
  • In Vitro
    Western Blot Analysis Cell Line:HEK293 cells Concentration:50 μM Incubation Time:Overnight Result:Partial rescued the total and surface expression of A432T.
  • In Vivo
    ——
  • Synonyms
    CBA | 4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    TRP/TRPV Channel
  • Recptor
    TRPM4
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    351424-20-9
  • Formula Weight
    340.16
  • Molecular Formula
    C15H11Cl2NO4
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:80mg/ml(235.18mM; need ultrasonic)
  • SMILES
    OC(c(ccc(Cl)c1)c1NC(COc(cccc1)c1Cl)=O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Ozhathil L C , Delalande C , Bianchi B , et al. Identification of potent and selective small molecule inhibitors of the cation channel TRPM4[J]. British Journal of Pharmacology, 2018.
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