TRPM4-IN-1( CBA | 4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid )

Catalog No. M24301 CAS No. 351424-20-9

TRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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Biological Information

Product Name

TRPM4-IN-1
Note

Research use only, not for human use.
Brief Description

TRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.
Description

TRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.
In Vitro

Western Blot Analysis Cell Line:HEK293 cells Concentration:50 μM Incubation Time:Overnight Result:Partial rescued the total and surface expression of A432T.
In Vivo

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Synonyms

CBA | 4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid
Pathway

Membrane Transporter/Ion Channel
Target

TRP/TRPV Channel
Recptor

TRPM4
Research Area

——
Indication

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Chemical Information

CAS Number

351424-20-9
Formula Weight

340.16
Molecular Formula

C15H11Cl2NO4
Purity

>98% (HPLC)
Solubility

DMSO:80mg/ml(235.18mM; need ultrasonic)
SMILES

OC(c(ccc(Cl)c1)c1NC(COc(cccc1)c1Cl)=O)=O
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Ozhathil L C , Delalande C , Bianchi B , et al. Identification of potent and selective small molecule inhibitors of the cation channel TRPM4[J]. British Journal of Pharmacology, 2018.

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