TMS
CAS No. 24144-92-1
TMS ( 2,3',4,5'-Tetramethoxystilbene )
Catalog No. M13695 CAS No. 24144-92-1
TMS is a very selective and potent competitive inhibitor of P450 1B1 (CYP1A1). It has strong selectivity among P450 family 1 enzymes.
Purity : >98%(HPLC)
Size | Price / USD | Stock | Quantity |
5MG | 42 | In Stock |
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10MG | 69 | In Stock |
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25MG | 138 | In Stock |
|
50MG | 251 | In Stock |
|
100MG | 374 | In Stock |
|
500MG | 848 | In Stock |
|
1G | Get Quote | In Stock |
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Biological Information
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Product NameTMS
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NoteResearch use only, not for human use.
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Brief DescriptionTMS is a very selective and potent competitive inhibitor of P450 1B1 (CYP1A1). It has strong selectivity among P450 family 1 enzymes.
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DescriptionTMS is a very selective and potent competitive inhibitor of P450 1B1 (CYP1A1). It has strong selectivity among P450 family 1 enzymes. TMS exhibits 50-fold selectivity for P450 1B1 over P4501A1 and 500-fold selectivity for P450 1B1 over P450 1A2.
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Synonyms2,3',4,5'-Tetramethoxystilbene
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PathwayMetabolic Enzyme/Protease
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TargetP450
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RecptorCYP450 1B1
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number24144-92-1
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Formula Weight300.35
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Molecular FormulaC18H20O4
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Purity>98%(HPLC)
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SolubilityDMSO:10 mM
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SMILESCOC1=CC(OC)=CC(/C=C/C2=CC=C(OC)C=C2OC)=C1
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Chemical Name(E)-1-(3,5-dimethoxystyryl)-2,4-dimethoxybenzene
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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Rhodionin
Rhodionin and rhodionin can inhibit cytochrome P450 2D6 non-competitively with high specificity which could have implications for interactions with co-administered drugs; they can significantly suppress the elevation of the postprandial blood triglyceride level suggests that they may be to the treatment of lifestyle-related diseases such as hyperlipidemia and exogeneous obesity and to health foods.
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2,6-Dimethylquinolin...
2,6-Dimethylquinoline is a natural product extracted from the roots of Peucedantu praeruptorum. 2,6-Dimethylquinoline is an inhibitor of CYP1A2 and CYP2B6 with an IC50 of 3.3 and 480 μM, respectively.
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Tienilic Acid
Tienilic Acid is a uricosuric diuretic with certain hepatotoxicity.