THIP
CAS No. 64603-91-4
THIP ( Gaboxadol; Gaboxadolum )
Catalog No. M26482 CAS No. 64603-91-4
THIP has a strong affinity for the δ subunit of GABAA receptors. THIP is a functionally selective GABAAR ligand, agonistic to α4β1δ, α4β3δ, and weakly antagonistic to αβγ and α4β2δ GABAARs.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 49 | Get Quote |
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Biological Information
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Product NameTHIP
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NoteResearch use only, not for human use.
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Brief DescriptionTHIP has a strong affinity for the δ subunit of GABAA receptors. THIP is a functionally selective GABAAR ligand, agonistic to α4β1δ, α4β3δ, and weakly antagonistic to αβγ and α4β2δ GABAARs.
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DescriptionTHIP has a strong affinity for the δ subunit of GABAA receptors. THIP is a functionally selective GABAAR ligand, agonistic to α4β1δ, α4β3δ, and weakly antagonistic to αβγ and α4β2δ GABAARs.
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SynonymsGaboxadol; Gaboxadolum
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PathwayOthers
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TargetOther Targets
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RecptorPPARγ
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Research Area——
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Indication——
Chemical Information
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CAS Number64603-91-4
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Formula Weight140.1
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Molecular FormulaC6H8N2O2
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Purity>98% (HPLC)
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Solubility——
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SMILESOc1noc2CNCCc12
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Rasmus K Petersen, et al. Pharmacophore-driven identification of PPARγ agonists from natural sources. J Comput Aided Mol Des. 2011 Feb;25(2):107-16.
molnova catalog
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