TC-G-1008

CAS No. 1621175-65-2

TC-G-1008 ( GPR39-C3, GPR39 C3, TC-G-1008, TCG1008, TCG 1008 )

Catalog No. M18094 CAS No. 1621175-65-2

TC-G-1008 is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively).

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 53 In Stock
5MG 83 In Stock
10MG 143 In Stock
25MG 303 In Stock
50MG 519 In Stock
100MG 746 In Stock
500MG 1512 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    TC-G-1008
  • Note
    Research use only, not for human use.
  • Brief Description
    TC-G-1008 is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively).
  • Description
    TC-G-1008, also known as GPR39-C3, is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively).
  • Synonyms
    GPR39-C3, GPR39 C3, TC-G-1008, TCG1008, TCG 1008
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    rat GPR39; human GPR39
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1621175-65-2
  • Formula Weight
    418.9
  • Molecular Formula
    C18H19ClN6O2S
  • Purity
    98%
  • Solubility
    DMSO : ≥ 100 mg/mL; 238.72 mM
  • SMILES
    CNc2nc(cc(NCc1ccc(NS(C)(=O)=O)cc1Cl)n2)c3ccccn3
  • Chemical Name
    N-[3-Chloro-4-[[[2-(methylamino)-6-(2-pyridinyl)-4-pyrimidinyl]amino]methyl]phenyl]methanesulfonamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Peukert S, et al. Discovery of 2-Pyridylpyrimidines as the First Orally Bioavailable GPR39 Agonists. ACS Med Chem Lett. 2014 Aug 4;5(10):1114-8.
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