Cart
sales@molnova.com
Home - Products - Others - Other Targets - Stiripentol

Stiripentol

CAS No. 49763-96-4

Stiripentol ( BCX2600 )

Catalog No. M18654 CAS No. 49763-96-4

Stiripentol (STP) is an anticonvulsant agent, which can inhibit N-demethylation of CLB to NCLB mediated by CYP3A4 (noncompetitively) and CYP2C19 (competitively) with Ki of 1.59/0.516 μM and IC50 of 1.58/3.29 μM, respectively.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 42 In Stock
10MG 68 In Stock
25MG 138 In Stock
50MG 195 In Stock
100MG 330 In Stock
200MG 489 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
Group Booking Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    Stiripentol
  • Note
    Research use only, not for human use.
  • Brief Description
    Stiripentol (STP) is an anticonvulsant agent, which can inhibit N-demethylation of CLB to NCLB mediated by CYP3A4 (noncompetitively) and CYP2C19 (competitively) with Ki of 1.59/0.516 μM and IC50 of 1.58/3.29 μM, respectively.
  • Description
    Stiripentol (STP) is an anticonvulsant agent, which can inhibit N-demethylation of CLB to NCLB mediated by CYP3A4 (noncompetitively) and CYP2C19 (competitively) with Ki of 1.59/0.516 μM and IC50 of 1.58/3.29 μM, respectively.
  • Synonyms
    BCX2600
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    CYP3A4; CYP2C19
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    49763-96-4
  • Formula Weight
    234.29
  • Molecular Formula
    C14H18O3
  • Purity
    98%
  • Solubility
    DMSO : 150 mg/mL 640.23 mM;
  • SMILES
    CC(C)(C)C(O)\C=C\c1ccc2OCOc2c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Giraud C, et al. In vitro and in vivo inhibitory effect of stiripentol on clobazam metabolism.Drug Metab Dispos. 2006 Apr;34(4):608-11. Epub 2006 Jan 13.
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • 5'-O-(4,4'-Dimethoxy...

    5'-O-(4,4'-Dimethoxytrityl)-2'-deoxyuridine is a competitive dUTP nucleotidohydrolase (dUTPase) inhibitor(Ki > 1 mM) in E. coli.

  • Depressine

    Depressine is a natural product from Gentiana depressa.

  • Boc-NH-PEG12-CH2CH2C...

    Boc-NH-PEG12-CH2CH2COOH is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs.

Sign In Join Free