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Stiripentol

CAS No. 49763-96-4

Stiripentol ( BCX2600 )

Catalog No. M18654 CAS No. 49763-96-4

Stiripentol (STP) is an anticonvulsant agent, which can inhibit N-demethylation of CLB to NCLB mediated by CYP3A4 (noncompetitively) and CYP2C19 (competitively) with Ki of 1.59/0.516 μM and IC50 of 1.58/3.29 μM, respectively.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Stiripentol
  • Note
    Research use only, not for human use.
  • Brief Description
    Stiripentol (STP) is an anticonvulsant agent, which can inhibit N-demethylation of CLB to NCLB mediated by CYP3A4 (noncompetitively) and CYP2C19 (competitively) with Ki of 1.59/0.516 μM and IC50 of 1.58/3.29 μM, respectively.
  • Description
    Stiripentol (STP) is an anticonvulsant agent, which can inhibit N-demethylation of CLB to NCLB mediated by CYP3A4 (noncompetitively) and CYP2C19 (competitively) with Ki of 1.59/0.516 μM and IC50 of 1.58/3.29 μM, respectively.
  • Synonyms
    BCX2600
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    CYP3A4; CYP2C19
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    49763-96-4
  • Formula Weight
    234.29
  • Molecular Formula
    C14H18O3
  • Purity
    98%
  • Solubility
    DMSO : 150 mg/mL 640.23 mM;
  • SMILES
    CC(C)(C)C(O)\C=C\c1ccc2OCOc2c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Giraud C, et al. In vitro and in vivo inhibitory effect of stiripentol on clobazam metabolism.Drug Metab Dispos. 2006 Apr;34(4):608-11. Epub 2006 Jan 13.
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