Setiptiline
CAS No. 57262-94-9
Setiptiline ( Teciptiline;Org-8282;MO-8282 )
Catalog No. M15088 CAS No. 57262-94-9
A tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
100MG | Get Quote | Get Quote |
|
200MG | Get Quote | Get Quote |
|
500MG | Get Quote | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameSetiptiline
-
NoteResearch use only, not for human use.
-
Brief DescriptionA tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist.
-
DescriptionA tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist, as well as an H1 receptor inverse agonist/antihistamine.Depression Approved
-
SynonymsTeciptiline;Org-8282;MO-8282
-
PathwayEndocrinology/Hormones
-
Target5-HT Receptor
-
Recptor5-HT Receptor
-
Research AreaNeurological Disease
-
IndicationDepression
Chemical Information
-
CAS Number57262-94-9
-
Formula Weight261.36
-
Molecular FormulaC19H19N
-
Purity>98% (HPLC)
-
Solubility10 mM in DMSO
-
SMILESCN1CCC2=C(C1)C3=CC=CC=C3CC4=CC=CC=C24
-
Chemical Name1H-Dibenzo[3,4:6,7]cyclohepta[1,2-c]pyridine, 2,3,4,9-tetrahydro-2-methyl-
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Niho T, et al. Nihon Yakurigaku Zasshi. 1986 Oct;88(4):309-20.
2. Mizota M, et al. Nihon Yakurigaku Zasshi. 1986 Dec;88(6):457-66.
3. Przegaliński E, et al. Pol J Pharmacol Pharm. 1986 Jul-Aug;38(4):377-84.
2. Mizota M, et al. Nihon Yakurigaku Zasshi. 1986 Dec;88(6):457-66.
3. Przegaliński E, et al. Pol J Pharmacol Pharm. 1986 Jul-Aug;38(4):377-84.
molnova catalog
related products
-
PRX-08066
PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.
-
RG2833
RG2833 (RGFP109), a brain-penetrant HDAC inhibitor, is with IC50 of 60 nM and 50 nM for HDAC1 and HDAC3, respectively.
-
Sumatriptan succinat...
Sumatriptan succinate is a serotonin1 (5-HT1) receptor agonist, which is effective in the acute treatment of migraine headache.