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Home - Products - Apoptosis - Adenosine Receptor - ST-4206

ST-4206

CAS No. 1246018-36-9

ST-4206( ST 4206 | ST4206 )

Catalog No. M10995 CAS No. 1246018-36-9

A metabolite of ST1535, which is potent, selective A2A adenosine receptor antagonist with Ki of 6.6 nM.

Purity : >98% (HPLC)

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Biological Information

  • Product Name
    ST-4206
  • Note
    Research use only, not for human use.
  • Brief Description
    A metabolite of ST1535, which is potent, selective A2A adenosine receptor antagonist with Ki of 6.6 nM.
  • Description
    A metabolite of ST1535, which is potent, selective A2A adenosine receptor antagonist with Ki of 6.6 nM.
  • In Vitro
    ST4206 inhibits agonist-induced cAMP accumulation with an IC50 of 990 nM.
  • In Vivo
    ST4206 (10, 20, and 40 mg/kg, p.o.) antagonizes haloperidol-induced catalepsy, and increases motor activity in a dose dependent manner in mice.ST4206 (20 and 40 mg/kg) significantly increases the number of contralateral turns induced by l-DOPA in rats. ST4206 is orally active at concentrations of 10, 20, and 40 mg/kg in haloperidol-induced catalepsy in mice.
  • Synonyms
    ST 4206 | ST4206
  • Pathway
    Apoptosis
  • Target
    Adenosine Receptor
  • Recptor
    Adenosine Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1246018-36-9
  • Formula Weight
    286.299
  • Molecular Formula
    C12H14N8O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CC(CCC1=NC(N)=C2N=C(N3N=CC=N3)N(C)C2=N1)=O
  • Chemical Name
    4-(6-amino-9-methyl-8-(2H-1,2,3-triazol-2-yl)-9H-purin-2-yl)butan-2-one

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Stasi MA, et al. Eur J Pharmacol. 2015 Aug 15;761:353-61.
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