
ST-4206
CAS No. 1246018-36-9
ST-4206( ST 4206 | ST4206 )
Catalog No. M10995 CAS No. 1246018-36-9
A metabolite of ST1535, which is potent, selective A2A adenosine receptor antagonist with Ki of 6.6 nM.
Purity : >98% (HPLC)






Size | Price / USD | Stock | Quantity |
5MG | 1053 | Get Quote |
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50MG | 2142 | Get Quote |
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100MG | 2790 | Get Quote |
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200MG | Get Quote | Get Quote |
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500MG | Get Quote | Get Quote |
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1G | Get Quote | Get Quote |
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Biological Information
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Product NameST-4206
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NoteResearch use only, not for human use.
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Brief DescriptionA metabolite of ST1535, which is potent, selective A2A adenosine receptor antagonist with Ki of 6.6 nM.
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DescriptionA metabolite of ST1535, which is potent, selective A2A adenosine receptor antagonist with Ki of 6.6 nM.
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In VitroST4206 inhibits agonist-induced cAMP accumulation with an IC50 of 990 nM.
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In VivoST4206 (10, 20, and 40 mg/kg, p.o.) antagonizes haloperidol-induced catalepsy, and increases motor activity in a dose dependent manner in mice.ST4206 (20 and 40 mg/kg) significantly increases the number of contralateral turns induced by l-DOPA in rats. ST4206 is orally active at concentrations of 10, 20, and 40 mg/kg in haloperidol-induced catalepsy in mice.
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SynonymsST 4206 | ST4206
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PathwayApoptosis
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TargetAdenosine Receptor
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RecptorAdenosine Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number1246018-36-9
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Formula Weight286.299
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Molecular FormulaC12H14N8O
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Purity>98% (HPLC)
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Solubility——
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SMILESCC(CCC1=NC(N)=C2N=C(N3N=CC=N3)N(C)C2=N1)=O
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Chemical Name4-(6-amino-9-methyl-8-(2H-1,2,3-triazol-2-yl)-9H-purin-2-yl)butan-2-one
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Stasi MA, et al. Eur J Pharmacol. 2015 Aug 15;761:353-61.
molnova catalog



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