SP-13786( UAMC-1110 )

Catalog No. M21138 CAS No. 1448440-52-5

SP-13786 is an inhibitor of fibroblast activation protein (FAP) (IC50 : 3.2 nM); also inhibits prolyl oligopeptidase (PREP) ( IC50 : 1.8 μM).

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
2MG	115	In Stock
5MG	191	In Stock
10MG	282	In Stock
25MG	475	In Stock
50MG	687	In Stock
100MG	963	In Stock
200MG	Get Quote	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

Group Booking Get Quotation Bulk Inquiry Add to Cart

Biological Information

Product Name

SP-13786
Note

Research use only, not for human use.
Brief Description

SP-13786 is an inhibitor of fibroblast activation protein (FAP) (IC50 : 3.2 nM); also inhibits prolyl oligopeptidase (PREP) ( IC50 : 1.8 μM).
Description

SP-13786 is an inhibitor of fibroblast activation protein (FAP) (IC50 : 3.2 nM); also inhibits prolyl oligopeptidase (PREP) ( IC50 : 1.8 μM).
In Vitro

——
In Vivo

——
Synonyms

UAMC-1110
Pathway

Others
Target

Other Targets
Recptor

FAP
Research Area

——
Indication

——

Chemical Information

CAS Number

1448440-52-5
Formula Weight

344.32
Molecular Formula

C17H14F2N4O2
Purity

>98% (HPLC)
Solubility

DMSO:100 mg/mL (290.43 mM; Need ultrasonic)
SMILES

N#CC1CC(F)(F)CN1C(=O)CNC(=O)c1ccnc2ccccc12
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Jansen K Heirbaut L Verkerk R et al. Extended Structure–Activity Relationship and Pharmacokinetic Investigation of (4-Quinolinoyl)glycyl-2-cyanopyrrolidine Inhibitors of Fibroblast Activation Protein (FAP)[J]. Journal of Medicinal Chemistry 2014 57(7):3053-3074.

Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog

Product			Quantity Required*
Name *			E-mail Address *
Organization *			Phone Number
Remarks