Cart
sales@molnova.com
Home - Products - Others - Other Targets - SGC-CBP30

SGC-CBP30

CAS No. 1613695-14-9

SGC-CBP30( SGC-CBP30 | SGC-CBP 30 | SGC-CBP-30 )

Catalog No. M17342 CAS No. 1613695-14-9

SGC-CBP30 is an effective CREBBP/EP300 inhibitor (IC50: 21/38 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 59 In Stock
5MG 72 In Stock
10MG 110 In Stock
25MG 200 In Stock
50MG 335 In Stock
100MG 500 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    SGC-CBP30
  • Note
    Research use only, not for human use.
  • Brief Description
    SGC-CBP30 is an effective CREBBP/EP300 inhibitor (IC50: 21/38 nM).
  • Description
    SGC-CBP30 is a potent and selective inhibitor of CREBBP (CBP) and EP300; which are general transcriptional co-activators. CREBBP has also been associated with Amyotrophic Lateral Sclerosis (ALS) or Lou Gehrig?’s disease, a neurodegenerative disease with progressive degeneration of motor neurons in the brain and spinal cord, Alzheimer's disease and poly glutamine repeat diseases such as Spinal and Bulbar Muscular Atrophy and Huntington?’s disease.
  • In Vitro
    ——
  • In Vivo
    Animal Model:Sprague-Dawley (SD) rats (aged 3-4 weeks) injected with NSC-125066 Dosage:25 mg/kg Administration:Oral administration; daily; for 14 days Result:Slightly alleviated alveolar bronchial fibrosis induced by NSC-125066.
  • Synonyms
    SGC-CBP30 | SGC-CBP 30 | SGC-CBP-30
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    CREBBP| EP300
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    1613695-14-9
  • Formula Weight
    509.04
  • Molecular Formula
    C28H33CIN4O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : ≥ 31 mg/mL; 60.90 mM
  • SMILES
    Cc1noc(C)c1c1cc2nc(CCc3ccc(OC)c(Cl)c3)n(C[C@H](C)N3CCOCC3)c2cc1
  • Chemical Name
    (S)-4-(1-(2-(3-chloro-4-methoxyphenethyl)-5-(3,5-dimethylisoxazol-4-yl)-1H-benzo[d]imidazol-1-yl)propan-2-yl)morpholine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Structural Genomics Consortium
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • Indecainide

    Indecainide (Ricainid) is a novel antiarrhythmic compound that is carcinogenic and can be used to study chronic stable ventricular arrhythmias secondary to coronary artery disease or cardiomyopathy.

  • (R)-Citronellol

    D-Citronellol is found in herbs and spices as well as bilberry. D-Citronellol is a constituent of black cumin (Nigella sativa) seeds. D-Citronellol is a common constituent of plant oils especially in the Rutaceae.

  • Carbetamide

    Carbetamide is a herbicide with a good reproduction of mobility in the soil.

Sign In Join Free