Rhapontigenin
CAS No. 500-65-2
Rhapontigenin ( —— )
Catalog No. M18663 CAS No. 500-65-2
Rhapontigenin is a mechanism-based, selective inactivator of cytochrome P450 1A1 (IC50: 400 nM), an aryl hydrocarbon hydroxylase which activates polycyclic aromatic hydrocarbons that act as procarcinogens.
Purity : 98%
Size | Price / USD | Stock | Quantity |
5MG | 88 | In Stock |
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10MG | 166 | In Stock |
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25MG | 321 | In Stock |
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50MG | 483 | In Stock |
|
100MG | 605 | In Stock |
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200MG | Get Quote | In Stock |
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500MG | Get Quote | In Stock |
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1G | Get Quote | In Stock |
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Biological Information
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Product NameRhapontigenin
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NoteResearch use only, not for human use.
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Brief DescriptionRhapontigenin is a mechanism-based, selective inactivator of cytochrome P450 1A1 (IC50: 400 nM), an aryl hydrocarbon hydroxylase which activates polycyclic aromatic hydrocarbons that act as procarcinogens.
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DescriptionRhapontigenin is a mechanism-based, selective inactivator of cytochrome P450 1A1 (IC50: 400 nM), an aryl hydrocarbon hydroxylase which activates polycyclic aromatic hydrocarbons that act as procarcinogens. Rhapontigenin is a natural analog of resveratrol with antioxidant and anti-cancer activity. At higher concentrations, rhapontigenin inhibits the proliferation of HL-60R and HepG2 cancer cell lines (IC50: 48 μM).
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetAChR
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RecptorCYP1A1
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Research AreaOthers-Field
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Indication——
Chemical Information
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CAS Number500-65-2
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Formula Weight258.3
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Molecular FormulaC15H14O4
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Purity98%
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Solubility——
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SMILESCOc1c(cc(cc1)/C=C/c1cc(cc(c1)O)O)O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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Dinotefuran
Dinotefuran is an insecticide of the neonicotinoid class for control of insect pests such as aphids whiteflies thrips leafhoppers leafminers.?Its mechanism of action involves disruption of the insect's nervous system by inhibiting nicotinic acetylcholine receptors.
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GZD 824
GZD824 is an orally bioavailable Bcr-Abl inhibitor for Bcr-Abl(WT, IC50: 0.34 nM) and Bcr-Abl(T315I, IC50: 0.68 nM).
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Acetamiprid
Acetamiprid is a nicotinic acetylcholine receptor (nAChR) agonist. Acetamiprid is a neonicotinoid insecticide used worldwide. It is shown to be associated with neuromuscular and reproductive disorders. Acetamiprid decreases in body weight and mildly affected spermatogenesis.