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Relebactam
CAS No. 1174018-99-5
Relebactam ( MK-7655 )
Catalog No. M10588 CAS No. 1174018-99-5
Relebactam (MK-7655)is a novel β-lactamase inhibitor that inhibited both class A and C β-lactamases in vitro.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 87 | In Stock |
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| 10MG | 140 | In Stock |
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| 25MG | 260 | In Stock |
|
| 50MG | 484 | In Stock |
|
| 100MG | 700 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameRelebactam
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NoteResearch use only, not for human use.
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Brief DescriptionRelebactam (MK-7655)is a novel β-lactamase inhibitor that inhibited both class A and C β-lactamases in vitro.
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DescriptionRelebactam (MK-7655)is a novel β-lactamase inhibitor that inhibited both class A and C β-lactamases in vitro; effectively restored imipenem's activity against imipenem-resistant Pseudomonas and Klebsiella strains at clinically achievable concentrations; reduces imipenem MICs for Enterobacteriaceae with KPC carbapenemases from 16-64 mg/L to 0.12-1 mg/L at a concentration of 4 mg/L.Bacterial Infection Phase 3 Clinical
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SynonymsMK-7655
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PathwayGPCR/G Protein
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TargetAntibacterial
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Recptordiazabicyclooctane
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Research AreaInfection
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IndicationBacterial Infection
Chemical Information
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CAS Number1174018-99-5
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Formula Weight348.38
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Molecular FormulaC12H20N4O6S
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESO=S(O)(ON1[C@]2([H])CC[C@@H](C(NC3CCNCC3)=O)[N@@](C2)C1=O)=O
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Chemical NameSulfuric acid, mono[(1R,2S,5R)-7-oxo-2-[(4-piperidinylamino)carbonyl]-1,6-diazabicyclo[3.2.1]oct-6-yl] ester
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Hirsch EB, et al. Antimicrob Agents Chemother. 2012 Jul;56(7):3753-7.
2. Blizzard TA, et al. Bioorg Med Chem Lett. 2014 Feb 1;24(3):780-5.
3. Livermore DM, et al. J Antimicrob Chemother. 2013 Oct;68(10):2286-90.
2. Blizzard TA, et al. Bioorg Med Chem Lett. 2014 Feb 1;24(3):780-5.
3. Livermore DM, et al. J Antimicrob Chemother. 2013 Oct;68(10):2286-90.
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