Relebactam

CAS No. 1174018-99-5

Relebactam ( MK-7655 )

Catalog No. M10588 CAS No. 1174018-99-5

Relebactam (MK-7655)is a novel β-lactamase inhibitor that inhibited both class A and C β-lactamases in vitro.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 87 In Stock
10MG 140 In Stock
25MG 260 In Stock
50MG 484 In Stock
100MG 700 In Stock
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Biological Information

  • Product Name
    Relebactam
  • Note
    Research use only, not for human use.
  • Brief Description
    Relebactam (MK-7655)is a novel β-lactamase inhibitor that inhibited both class A and C β-lactamases in vitro.
  • Description
    Relebactam (MK-7655)is a novel β-lactamase inhibitor that inhibited both class A and C β-lactamases in vitro; effectively restored imipenem's activity against imipenem-resistant Pseudomonas and Klebsiella strains at clinically achievable concentrations; reduces imipenem MICs for Enterobacteriaceae with KPC carbapenemases from 16-64 mg/L to 0.12-1 mg/L at a concentration of 4 mg/L.Bacterial Infection Phase 3 Clinical
  • Synonyms
    MK-7655
  • Pathway
    GPCR/G Protein
  • Target
    Antibacterial
  • Recptor
    diazabicyclooctane
  • Research Area
    Infection
  • Indication
    Bacterial Infection

Chemical Information

  • CAS Number
    1174018-99-5
  • Formula Weight
    348.38
  • Molecular Formula
    C12H20N4O6S
  • Purity
    >98% (HPLC)
  • Solubility
    10 mM in DMSO
  • SMILES
    O=S(O)(ON1[C@]2([H])CC[C@@H](C(NC3CCNCC3)=O)[N@@](C2)C1=O)=O
  • Chemical Name
    Sulfuric acid, mono[(1R,2S,5R)-7-oxo-2-[(4-piperidinylamino)carbonyl]-1,6-diazabicyclo[3.2.1]oct-6-yl] ester

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Hirsch EB, et al. Antimicrob Agents Chemother. 2012 Jul;56(7):3753-7.
2. Blizzard TA, et al. Bioorg Med Chem Lett. 2014 Feb 1;24(3):780-5.
3. Livermore DM, et al. J Antimicrob Chemother. 2013 Oct;68(10):2286-90.
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