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Ralinepag
CAS No. 1187856-49-0
Ralinepag ( APD811 )
Catalog No. M17861 CAS No. 1187856-49-0
Ralinepag is a potent, orally bioavailable and non-prostanoid prostacyclin (IP) receptor agonist, with EC50s of 8.5 nM, 530 nM and 850 nM for human and rat IP receptor and human DP1 receptor, respectively.
Purity : 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 120 | In Stock |
|
| 10MG | 215 | In Stock |
|
| 25MG | 315 | In Stock |
|
| 50MG | 471 | In Stock |
|
| 100MG | 683 | In Stock |
|
| 500MG | 1422 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameRalinepag
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NoteResearch use only, not for human use.
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Brief DescriptionRalinepag is a potent, orally bioavailable and non-prostanoid prostacyclin (IP) receptor agonist, with EC50s of 8.5 nM, 530 nM and 850 nM for human and rat IP receptor and human DP1 receptor, respectively.
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DescriptionRalinepag is a potent, orally bioavailable and non-prostanoid prostacyclin (IP) receptor agonist, with EC50s of 8.5 nM, 530 nM and 850 nM for human and rat IP receptor and human DP1 receptor, respectively.
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SynonymsAPD811
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PathwayOthers
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TargetOther Targets
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RecptorProstacyclin receptor
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Research AreaOthers-Field
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Indication——
Chemical Information
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CAS Number1187856-49-0
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Formula Weight431.91
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Molecular FormulaC23H26ClNO5
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Purity98%
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SolubilityDMSO : 125 mg/mL 289.41 mM;
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SMILESClc1ccc(cc1)N(c2ccccc2)C(=O)OC[C@H]3CC[C@H](COCC(=O)O)CC3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Tran TA, et al. J Med Chem. 2017 Feb 9;60(3):913-927
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