RO5454291

CAS No.

RO5454291 ( RO 5454291 )

Catalog No. M16939 CAS No.

RO5258638 is a small molecule inhibitor of CDK5-p25 protein-protein interaction with IC50 of 1.39 uM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    RO5454291
  • Note
    Research use only, not for human use.
  • Brief Description
    RO5258638 is a small molecule inhibitor of CDK5-p25 protein-protein interaction with IC50 of 1.39 uM.
  • Description
    RO5258638 is a small molecule inhibitor of CDK5-p25 protein-protein interaction with IC50 of 1.39 uM.
  • Synonyms
    RO 5454291
  • Pathway
    Angiogenesis
  • Target
    CDK
  • Recptor
    CDK
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    --
  • Formula Weight
    357.46
  • Molecular Formula
    C19H27N5O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CCC(C)(C)C(N(C1)CC2=C1C(NC3=NC(OC)=CC=C3)=NN2)=O
  • Chemical Name
    1-(3-((6-methoxypyridin-2-yl)amino)-6,6-dimethyl-4,6-dihydropyrrolo[3,4-c]pyrazol-5(1H)-yl)-2,2-dimethylbutan-1-one

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Bellón-Echeverría I, et al. Sci Rep. 2018 Mar 23;8(1):5083.
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