RO5258638

CAS No.

RO5258638 ( RO 5258638 )

Catalog No. M16937 CAS No.

RO5258638 is a small molecule inhibitor of CDK5-p25 protein-protein interaction.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    RO5258638
  • Note
    Research use only, not for human use.
  • Brief Description
    RO5258638 is a small molecule inhibitor of CDK5-p25 protein-protein interaction.
  • Description
    RO5258638 is a small molecule inhibitor of CDK5-p25 protein-protein interaction.
  • Synonyms
    RO 5258638
  • Pathway
    Angiogenesis
  • Target
    CDK
  • Recptor
    CDK
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    --
  • Formula Weight
    396.47
  • Molecular Formula
    C19H20N6O2S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    N#CC1=CN(C2=NC(NC3CCN(S(=O)(C)=O)CC3)=NC=C2)C4=C1C=CC=C4
  • Chemical Name
    1-(2-((1-(methylsulfonyl)piperidin-4-yl)amino)pyrimidin-4-yl)-1H-indole-3-carbonitrile

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Bellón-Echeverría I, et al. Sci Rep. 2018 Mar 23;8(1):5083.
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