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RHPS4
CAS No. 390362-78-4
RHPS4( —— )
Catalog No. M17501 CAS No. 390362-78-4
RHPS4 is a potent inhibitor of Telomerase at submicromolar.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 35 | Get Quote |
|
| 10MG | 58 | Get Quote |
|
| 25MG | 113 | Get Quote |
|
| 50MG | 215 | Get Quote |
|
| 100MG | 356 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameRHPS4
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NoteResearch use only, not for human use.
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Brief DescriptionRHPS4 is a potent inhibitor of Telomerase at submicromolar.
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DescriptionRHPS4 is a potent inhibitor of Telomerase at submicromolar.
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In VitroCell Proliferation Assay Cell Line:MCF-7, MCF-7 vector control, and MCF-7 c81 cells.Concentration:0, 0.2, 0.5, or 1 μM.Incubation Time:7 days.Result:Inhibited cell proliferation.
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In VivoAnimal Model:CD-1 male nude (nu/nu) mice, 6–8 weeks old and weighing 22-24 g (H460, CG5 and HT29, PC3 and M14 cancer models).Dosage:15 mg/kg.Administration:IV, daily for 15 consecutive days.Result:Active as a single agent on all the tumors analyzed. CG5 breast xenografts resulted in the most sensitive tumor.
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Synonyms——
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PathwayPI3K/Akt/mTOR signaling
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TargetGSK-3
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RecptorTelomerase
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number390362-78-4
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Formula Weight458.48
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Molecular FormulaC22H17F2N2·CH3O4S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 1 mg/mL (2.18 mM)
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SMILESCC1=CC2=C3C(=C1)C4=C(C=CC(=C4)F)[N+](=C3C5=C(N2C)C=CC(=C5)F)C.COS(=O)(=O)[O-]
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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