Prucalopride

CAS No. 179474-81-8

Prucalopride ( Prucalopride; Prucalopride free base )

Catalog No. M12708 CAS No. 179474-81-8

Prucalopride is a selective, high affinity 5-HT receptor agonist for 5-HT4A and 5-HT4B receptor with Ki of 2.5 nM and 8 nM, respectively.

Purity : >98%(HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 29 Get Quote
10MG 47 Get Quote
25MG 61 Get Quote
50MG 73 Get Quote
100MG 126 Get Quote
200MG 178 Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Prucalopride
  • Note
    Research use only, not for human use.
  • Brief Description
    Prucalopride is a selective, high affinity 5-HT receptor agonist for 5-HT4A and 5-HT4B receptor with Ki of 2.5 nM and 8 nM, respectively.
  • Description
    Prucalopride is a selective, high affinity 5-HT receptor agonist for 5-HT4A and 5-HT4B receptor with Ki of 2.5 nM and 8 nM, respectively, exhibits >290-fold selectivity against other 5-HT receptor subtypes.
  • Synonyms
    Prucalopride; Prucalopride free base
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT1A; 5-HT1B; 5-HT3; 5-HT4A; 5-HT4B
  • Research Area
    Neurological Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    179474-81-8
  • Formula Weight
    367.87
  • Molecular Formula
    C18H26ClN3O3
  • Purity
    >98%(HPLC)
  • Solubility
    Ethanol: 38 mg/mL (103.29 mM); DMSO: 60 mg/mL (163.1 mM)
  • SMILES
    ClC1=CC(C(NC2CCN(CCCOC)CC2)=O)=C3C(CCO3)=C1N
  • Chemical Name
    4-amino-5-chloro-N-(1-(3-methoxypropyl)piperidin-4-yl)-2,3-dihydrobenzofuran-7-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Briejer MR, et al. Eur J Pharmacol, 2001, 423(1), 71-83.
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