Perlapine ( AW-14233;HF-2333;Hypnodine )

Catalog No. M13091 CAS No. 1977-11-3

Perlapine (AW-14233;HF-2333;Hypnodine) is a potent antihistamine that has high affinity for dopamine D1, α1, α2 and 5-HT2A receptors.

Purity : >98% (HPLC)

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Biological Information

Product Name

Perlapine
Note

Research use only, not for human use.
Brief Description

Perlapine (AW-14233;HF-2333;Hypnodine) is a potent antihistamine that has high affinity for dopamine D1, α1, α2 and 5-HT2A receptors.
Description

Perlapine (AW-14233;HF-2333;Hypnodine) is a potent antihistamine that has high affinity for dopamine D1, α1, α2 and 5-HT2A receptors with IC50 of 198, 19, 4945 and 70 nM, respectively; also has anticholinergic, antiserotonergic, antiadrenergic and antidopaminergic activity; also is a highly potent hM3Dq agonist (EC50=2.8 nM) but do not activate the native human M3 receptor (hM3, EC50>30 uM).
Synonyms

AW-14233;HF-2333;Hypnodine
Pathway

Endocrinology/Hormones
Target

5-HT Receptor
Recptor

5-HT Receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

1977-11-3
Formula Weight

291.40
Molecular Formula

C19H21N3
Purity

>98% (HPLC)
Solubility

——
SMILES

CN1CCN(C2=NC3=CC=CC=C3CC4=CC=CC=C42)CC1
Chemical Name

6-(4-Methyl-1-piperazinyl)-11H-dibenz[b,e]azepine

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Stille G, et al. Psychopharmacologia. 1973 Feb 20;28(4):325-37.
2. Wilk S, et al. Eur J Pharmacol. 1977 Jan 7;41(1):65-72.
3. Chen X, et al. ACS Chem Neurosci. 2015 Mar 18;6(3):476-84.

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