Parsaclisib
CAS No. 1426698-88-5
Parsaclisib ( INCB050465 )
Catalog No. M23581 CAS No. 1426698-88-5
Parsaclisib is a potent and selective inhibitor of PI3Kδ(IC50 of 1 nM at 1 mM ATP).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 290 | In Stock |
|
10MG | 470 | In Stock |
|
25MG | 763 | In Stock |
|
50MG | 1053 | In Stock |
|
100MG | 1422 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
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Product NameParsaclisib
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NoteResearch use only, not for human use.
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Brief DescriptionParsaclisib is a potent and selective inhibitor of PI3Kδ(IC50 of 1 nM at 1 mM ATP).
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DescriptionParsaclisib is a potent and selective inhibitor of PI3Kδ(IC50 of 1 nM at 1 mM ATP).
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SynonymsINCB050465
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PathwayPI3K/Akt/mTOR signaling
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TargetPI3K
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RecptorPI3Kδ
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Research Area——
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Indication——
Chemical Information
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CAS Number1426698-88-5
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Formula Weight432.9
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Molecular FormulaC20H22ClFN6O2
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Purity>98% (HPLC)
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SolubilityDMSO:122 mg/mL?(281.83 mM;?Need ultrasonic)
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SMILESCCOc(c([C@H](C)n1nc(C)c2c(N)ncnc12)c1)c([C@@H](C2)CNC2=O)c(F)c1Cl
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Niu Shin, et al. Abstract 2671: INCB050465, a novel PI3Kδ inhibitor, synergizes with PIM protein kinase inhibition to cause tumor regression in a model of DLBCL. Cancer Research. 2015, Aug. 75(15).
molnova catalog
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