Parsaclisib

CAS No. 1426698-88-5

Parsaclisib ( INCB050465 )

Catalog No. M23581 CAS No. 1426698-88-5

Parsaclisib is a potent and selective inhibitor of PI3Kδ(IC50 of 1 nM at 1 mM ATP).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 290 In Stock
10MG 470 In Stock
25MG 763 In Stock
50MG 1053 In Stock
100MG 1422 In Stock
200MG Get Quote In Stock
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Biological Information

  • Product Name
    Parsaclisib
  • Note
    Research use only, not for human use.
  • Brief Description
    Parsaclisib is a potent and selective inhibitor of PI3Kδ(IC50 of 1 nM at 1 mM ATP).
  • Description
    Parsaclisib is a potent and selective inhibitor of PI3Kδ(IC50 of 1 nM at 1 mM ATP).
  • Synonyms
    INCB050465
  • Pathway
    PI3K/Akt/mTOR signaling
  • Target
    PI3K
  • Recptor
    PI3Kδ
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1426698-88-5
  • Formula Weight
    432.9
  • Molecular Formula
    C20H22ClFN6O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:122 mg/mL?(281.83 mM;?Need ultrasonic)
  • SMILES
    CCOc(c([C@H](C)n1nc(C)c2c(N)ncnc12)c1)c([C@@H](C2)CNC2=O)c(F)c1Cl
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Niu Shin, et al. Abstract 2671: INCB050465, a novel PI3Kδ inhibitor, synergizes with PIM protein kinase inhibition to cause tumor regression in a model of DLBCL. Cancer Research. 2015, Aug. 75(15).
molnova catalog
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