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PU23
CAS No. 817635-93-1
PU23( —— )
Catalog No. M29003 CAS No. 817635-93-1
PU 23 is an inhibitor of multidrug-resistant protein 4 (MRP4).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 72 | Get Quote |
|
| 10MG | 115 | Get Quote |
|
| 25MG | 248 | Get Quote |
|
| 50MG | 393 | Get Quote |
|
| 100MG | 581 | Get Quote |
|
| 500MG | 1242 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NamePU23
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NoteResearch use only, not for human use.
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Brief DescriptionPU 23 is an inhibitor of multidrug-resistant protein 4 (MRP4).
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DescriptionPU 23 is an inhibitor of multidrug-resistant protein 4 (MRP4).(In Vitro):6-Mercaptopurine (6-MP) inhibits HEK293 and HEK293/MRP4 cells with IC50s of 2.81 and 14.11 μM, respectively. The combination of PU23 and 6-MP inhibits HEK293 and HEK293/MRP4 cells with IC50s of 1.84 and 6.06 μM, respectively.Preincubation of HEK293/MRP4 cells with PU 23 (50 μM) for 2 h also significantly increases the amount of 6-MP in cells .
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In Vitro6-Mercaptopurine (6-MP) inhibits HEK293 and HEK293/MRP4 cells with IC50s of 2.81 and 14.11 μM, respectively. The combination of PU 23 (Cpd23) and 6-Mercaptopurine (6-MP) inhibits HEK293 and HEK293/MRP4 cells with IC50s of 1.84 and 6.06 μM, respectively.Preincubation of HEK293/MRP4 cells with PU 23 (50 μM) for 2 h also significantly increases the amount of 6-MP in cells.
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In Vivo——
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetMRP
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RecptorMRP
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Research Area——
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Indication——
Chemical Information
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CAS Number817635-93-1
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Formula Weight425.52
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Molecular FormulaC21H19N3O3S2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (293.76 mM)
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SMILESO=C(NC(=S)NC1=CC=C(C=C1)S(=O)(=O)NCC1=CC=CC=C1)C1=CC=CC=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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