PTP1B-IN-1

CAS No. 612530-44-6

PTP1B-IN-1 ( PTP1B inhibitor )

Catalog No. M20750 CAS No. 612530-44-6

PTP1B-IN-1 is a potent inhibitor of protein tyrosine phosphatase 1B (PTP1B) (IC50 : 1.6 mM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 168 In Stock
5MG 262 In Stock
10MG 374 In Stock
25MG 623 In Stock
50MG 887 In Stock
100MG 1197 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    PTP1B-IN-1
  • Note
    Research use only not for human use.
  • Brief Description
    PTP1B-IN-1 is a potent inhibitor of protein tyrosine phosphatase 1B (PTP1B) (IC50 : 1.6 mM).
  • Description
    PTP1B-IN-1 is a potent inhibitor of protein tyrosine phosphatase 1B (PTP1B) (IC50 : 1.6 mM)
  • Synonyms
    PTP1B inhibitor
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Phosphatase
  • Recptor
    PTP1B
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    612530-44-6
  • Formula Weight
    212.23
  • Molecular Formula
    C8H8N2O3S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:38 mg/mL (179.05 mM)
  • SMILES
    O=C1CN(c2ccccc2)S(=O)(=O)N1
  • Chemical Name
    11-Dioxo-5-phenyl-125-thiadiazolidin-3-one

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Wang Y Yan F Ye Q et al. PTP1B inhibitor promotes endothelial cell motility by activating the DOCK180/Rac1 pathway[J]. Scientific Reports 2016 6:24111.
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