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Home - Products - Membrane Transporter/Ion Channel - GAT - PK-14105

PK-14105

CAS No. 107257-28-3

PK-14105( PK14105 )

Catalog No. M10296 CAS No. 107257-28-3

A potent photoaffinity ligand for the peripheral-type benzodiazepine binding site with Ki of 4 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    PK-14105
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent photoaffinity ligand for the peripheral-type benzodiazepine binding site with Ki of 4 nM.
  • Description
    A potent photoaffinity ligand for the peripheral-type benzodiazepine binding site with Ki of 4 nM; attaches covalently and specifically to all the PBS when cardiac membranes are irradiated with this compound under ultraviolet light.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    PK14105
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    GAT
  • Recptor
    GAT
  • Research Area
    Other Indications
  • Indication
    ——

Chemical Information

  • CAS Number
    107257-28-3
  • Formula Weight
    381.4002
  • Molecular Formula
    C21H20FN3O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥ 30 mg/mL
  • SMILES
    O=C(C1=CC2=C(C(C3=CC([N+]([O-])=O)=CC=C3F)=N1)C=CC=C2)N(C(CC)C)C
  • Chemical Name
    3-Isoquinolinecarboxamide, 1-(2-fluoro-5-nitrophenyl)-N-methyl-N-(1-methylpropyl)-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Doble A, et al. Mol Pharmacol. 1987 Jan;31(1):42-9. 2. Doble A, et al. J Recept Res. 1987;7(1-4):55-70. 3. Skowroński R, et al. Eur J Pharmacol. 1988 Mar 29;148(2):187-93.
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