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Home - Products - GPCR/G Protein - Melanocortin Receptor - PF-07258669

PF-07258669

CAS No. 2755890-53-8

PF-07258669( —— )

Catalog No. M36282 CAS No. 2755890-53-8

PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    PF-07258669
  • Note
    Research use only, not for human use.
  • Brief Description
    PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.
  • Description
    PF-07258669 is a melanocortin-4 receptor (MC4) antagonist. PF-07258669 can be used for the research of cachexia, anorexia, or anorexia nervosa.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Melanocortin Receptor
  • Recptor
    Melanocortin Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2755890-53-8
  • Formula Weight
    462.52
  • Molecular Formula
    C25H27FN6O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C([C@H](C)C=1C=C(OC)N=CC1F)(=O)N2C[C@@]3(NC=4C(CC3)=CC(=C(C)N4)C=5N=CC=CN5)CC2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Christopher Ryan BUTLER, et al. Spiro compounds as melanocortin 4 receptor antagonists and uses thereof. Patent. WO2021250541A1.
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