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PF-01247324

CAS No. 875051-72-2

PF-01247324 ( PF-01247324; PF 01247324; PF01247324 )

Catalog No. M19208 CAS No. 875051-72-2

PF-01247324 is a selective and orally bioavailable Nav1.8 channel blocker (IC50: 196 nM).

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    PF-01247324
  • Note
    Research use only, not for human use.
  • Brief Description
    PF-01247324 is a selective and orally bioavailable Nav1.8 channel blocker (IC50: 196 nM).
  • Description
    PF-01247324 is a novel selective and orally bioavailable Nav 1.8 channel blocker, attenuates nociception and sensory neuron excitability.
  • Synonyms
    PF-01247324; PF 01247324; PF01247324
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    Na(V1.8) channel
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    875051-72-2
  • Formula Weight
    330.6
  • Molecular Formula
    C13H10Cl3N3O
  • Purity
    98%
  • Solubility
    DMSO : ≥ 30 mg/mL; 90.74 mM
  • SMILES
    CNC(=O)c1ccc(c(N)n1)-c1cc(Cl)cc(Cl)c1Cl
  • Chemical Name
    6-amino-N-methyl-5-(2,3,5-trichlorophenyl)pyridine-2-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Payne CE, et al. A novel selective and orally bioavailable Nav 1.8 channel blocker, PF-01247324, attenuates nociception and sensory neuron excitability. Br J Pharmacol. 2015 May;172(10):2654-70.
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