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Home - Products - GPCR/G Protein - Antibacterial - P516-0475

P516-0475

CAS No. 1359627-33-0

P516-0475( P516-0475 | P5160475 | P516 0475 )

Catalog No. M11475 CAS No. 1359627-33-0

P516-0475 is a novel chemical inducer of Streptococcus quorum sensing acts by inhibiting the pheromone-degrading endopeptidase PepO (IC50=10 uM).

Purity : >98% (HPLC)

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Biological Information

  • Product Name
    P516-0475
  • Note
    Research use only, not for human use.
  • Brief Description
    P516-0475 is a novel chemical inducer of Streptococcus quorum sensing acts by inhibiting the pheromone-degrading endopeptidase PepO (IC50=10 uM).
  • Description
    P516-0475 is a novel chemical inducer of Streptococcus quorum sensing acts by inhibiting the pheromone-degrading endopeptidase PepO (IC50=10 uM); specifically induces expression of Rgg2/3-regulated genes in the presence of SHP pheromones at concentrations lower than typically required for QS induction; P516-0475 directly inhibits recombinant PepO in vitro as an uncompetitive inhibitor, induces QS by stabilizing SHP pheromones in culture.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    P516-0475 | P5160475 | P516 0475
  • Pathway
    GPCR/G Protein
  • Target
    Antibacterial
  • Recptor
    Antibacterial
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1359627-33-0
  • Formula Weight
    315.333
  • Molecular Formula
    C15H17N5O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C(C1=C2N(N=N1)C3=C(C=C(C)C=C3)NC2=O)NCCCOC
  • Chemical Name
    N-(3-methoxypropyl)-7-methyl-4-oxo-4,5-dihydro-[1,2,3]triazolo[1,5-a]quinoxaline-3-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Pérez Morales TG, et al. J Biol Chem. 2018 Jan 19;293(3):931-940.
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