Home - Products - Endocrinology/Hormones - 5-HT Receptor - Ogerin

Ogerin

CAS No. 1309198-71-7

Ogerin ( —— )

Catalog No. M23467 CAS No. 1309198-71-7

Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
2MG	40	In Stock
5MG	61	In Stock
10MG	105	In Stock
25MG	215	In Stock
50MG	361	In Stock
100MG	537	In Stock
200MG	Get Quote	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

Group Booking Get Quotation Bulk Inquiry Add to Cart

Biological Information

Product Name

Ogerin
Note

Research use only, not for human use.
Brief Description

Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice.
Description

Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice. Ogerin displays inverse agonist and antagonist activity (Ki, 220 nM) at A2A receptor and weak antagonist activity (Ki, 736 nM) at 5-HT2B receptor.
Synonyms

——
Pathway

Endocrinology/Hormones
Target

5-HT Receptor
Recptor

5-HT2B;A2A;GPR68
Research Area

——
Indication

——

Chemical Information

CAS Number

1309198-71-7
Formula Weight

307.4
Molecular Formula

C17H17N5O
Purity

>98% (HPLC)
Solubility

DMSO:250 mg/mL (813.40 mM; Need ultrasonic)
SMILES

OCC1=C(C2=NC(N)=NC(NCC3=CC=CC=C3)=N2)C=CC=C1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Huang XP, et al. Allosteric ligands for the pharmacologically dark receptors GPR68 and GPR65. Nature. 2015 Nov 26;527(7579):477-83.

Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog

related products

RS 127445

RS 127445 is a selective high affinity orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).
AC-90179 HCl

AC-90179 HCl is a selective inverse agonist of 5-HT2A receptor. AC-90179 HCl is an atypical antipsychotic pharmaceutical and has been shown to alleviate hallucinogen-induced vasocontriction.
glucosylvitexin

Glucosylvitexin inhibits TPO activity.

Sign In Join Free