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Ogerin
CAS No. 1309198-71-7
Ogerin ( —— )
Catalog No. M23467 CAS No. 1309198-71-7
Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 40 | In Stock |
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| 5MG | 61 | In Stock |
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| 10MG | 105 | In Stock |
|
| 25MG | 215 | In Stock |
|
| 50MG | 361 | In Stock |
|
| 100MG | 537 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameOgerin
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NoteResearch use only, not for human use.
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Brief DescriptionOgerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice.
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DescriptionOgerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice. Ogerin displays inverse agonist and antagonist activity (Ki, 220 nM) at A2A receptor and weak antagonist activity (Ki, 736 nM) at 5-HT2B receptor.
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Synonyms——
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT2B;A2A;GPR68
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Research Area——
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Indication——
Chemical Information
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CAS Number1309198-71-7
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Formula Weight307.4
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Molecular FormulaC17H17N5O
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Purity>98% (HPLC)
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SolubilityDMSO:250 mg/mL (813.40 mM; Need ultrasonic)
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SMILESOCC1=C(C2=NC(N)=NC(NCC3=CC=CC=C3)=N2)C=CC=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Huang XP, et al. Allosteric ligands for the pharmacologically dark receptors GPR68 and GPR65. Nature. 2015 Nov 26;527(7579):477-83.
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