Cart
sales@molnova.com
Ocinaplon
CAS No. 96604-21-6
Ocinaplon ( DOV 273547 )
Catalog No. M27674 CAS No. 96604-21-6
Ocinaplon is a GABAA receptors modulator.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 80 | Get Quote |
|
| 10MG | 140 | Get Quote |
|
| 25MG | 282 | Get Quote |
|
| 50MG | 421 | Get Quote |
|
| 100MG | 606 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameOcinaplon
-
NoteResearch use only, not for human use.
-
Brief DescriptionOcinaplon is a GABAA receptors modulator.
-
DescriptionOcinaplon is a GABAA receptors modulator.(In Vivo):In rats, ocinaplon produces significant muscle relaxation, ataxia, and sedation only at doses >25-fold higher than the minimum effective dose (3.1 mg/kg) in the Vogel "conflict" test.
-
SynonymsDOV 273547
-
PathwayOthers
-
TargetOther Targets
-
RecptorP2X7
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number96604-21-6
-
Formula Weight301.3
-
Molecular FormulaC17H11N5O
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESO=C(c1cnn2c(ccnc12)-c1ccncc1)c1ccccn1
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Hopper AT, et al. Synthesis and Characterization of the Novel Rodent-Active and CNS-Penetrant P2X7 Receptor Antagonist Lu AF27139. J Med Chem. 2021;64(8):4891-4902.
molnova catalog
related products
-
CFT7455
CFT7455 is an anti-cancer agent showing high affinity to the cereblon E3 ligase with a Kd of 0.9 nM. CFT7455 is an orally active degrader of zinc finger transcription factors Ikaros (IKZF1), and Aiolos (IKZF3).
-
TAK-981
TAK-981 is a selective the SUMOylation enzymatic cascade inhibitor, has potential immune-activating and antineoplastic activities.
-
GT 949
GT 949 is a selective excitatory positive allosteric modulator of amino acid transporter-2 (EAAT2) (EC50: 0.26 nM).
