Ocinaplon

CAS No. 96604-21-6

Ocinaplon ( DOV 273547 )

Catalog No. M27674 CAS No. 96604-21-6

Ocinaplon is a GABAA receptors modulator.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 80 Get Quote
10MG 140 Get Quote
25MG 282 Get Quote
50MG 421 Get Quote
100MG 606 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Ocinaplon
  • Note
    Research use only, not for human use.
  • Brief Description
    Ocinaplon is a GABAA receptors modulator.
  • Description
    Ocinaplon is a GABAA receptors modulator.(In Vivo):In rats, ocinaplon produces significant muscle relaxation, ataxia, and sedation only at doses >25-fold higher than the minimum effective dose (3.1 mg/kg) in the Vogel "conflict" test.
  • Synonyms
    DOV 273547
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    P2X7
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    96604-21-6
  • Formula Weight
    301.3
  • Molecular Formula
    C17H11N5O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C(c1cnn2c(ccnc12)-c1ccncc1)c1ccccn1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Hopper AT, et al. Synthesis and Characterization of the Novel Rodent-Active and CNS-Penetrant P2X7 Receptor Antagonist Lu AF27139. J Med Chem. 2021;64(8):4891-4902.
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