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Obicetrapib

CAS No. 866399-87-3

Obicetrapib( AMG-899 | AMG899 | TA-8995 | DEX-001 )

Catalog No. M16296 CAS No. 866399-87-3

Obicetrapib (AMG-899, TA-8995, DEX-001) is a potent, ora cholesteryl ester transfer protein (CETP) inhibitor for treatment of dyslipidaemia.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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2MG 264 Get Quote
5MG 403 Get Quote
10MG 592 Get Quote
25MG 888 Get Quote
50MG 1242 Get Quote
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Biological Information

  • Product Name
    Obicetrapib
  • Note
    Research use only, not for human use.
  • Brief Description
    Obicetrapib (AMG-899, TA-8995, DEX-001) is a potent, ora cholesteryl ester transfer protein (CETP) inhibitor for treatment of dyslipidaemia.
  • Description
    Obicetrapib (AMG-899, TA-8995, DEX-001) is a potent, ora cholesteryl ester transfer protein (CETP) inhibitor for treatment of dyslipidaemia.Dyslipidemia Phase 2 Clinical.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    AMG-899 | AMG899 | TA-8995 | DEX-001
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    CETP
  • Recptor
    CETP
  • Research Area
    Cardiovascular Disease
  • Indication
    Dyslipidemia

Chemical Information

  • CAS Number
    866399-87-3
  • Formula Weight
    722.609
  • Molecular Formula
    C32H31F9N4O5
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CCC1CC(C2=C(N1C(=O)OCC)C=CC(=C2)C(F)(F)F)N(CC3=CC(=CC(=C3)C(F)(F)F)C(F)(F)F)C4=NC=C(C=N4)OCCCC(=O)O
  • Chemical Name
    4-[2-[[3,5-bis(trifluoromethyl)phenyl]methyl-[(2R,4S)-1-ethoxycarbonyl-2-ethyl-6-(trifluoromethyl)-3,4-dihydro-2H-quinolin-4-yl]amino]pyrimidin-5-yl]oxybutanoic acid

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Ford J, et al. Br J Clin Pharmacol. 2014 Sep;78(3):498-508. 2. Hovingh GK, et al. Lancet. 2015 Aug 1;386(9992):452-60.
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