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NPAS3-IN-1

CAS No. 2207-44-5

NPAS3-IN-1( —— )

Catalog No. M37303 CAS No. 2207-44-5

NPAS3-IN-1 is a potent inhibitor of NPAS3-ARNT heterodimerization, modulating NPAS3 transcription by targeting the interaction between NPAS3 and ARNT at the cellular level.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Biological Information

Product Name

NPAS3-IN-1
Note

Research use only, not for human use.
Brief Description

NPAS3-IN-1 is a potent inhibitor of NPAS3-ARNT heterodimerization, modulating NPAS3 transcription by targeting the interaction between NPAS3 and ARNT at the cellular level.
Description

NPAS3-IN-1 is a potent inhibitor of NPAS3-ARNT heterodimerization and regulates NPAS3 transcription by disrupting the heterodimerization of NPAS3 with ARNT at the cellular level.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Others
Target

Other Targets
Recptor

Others
Research Area

——
Indication

——

Chemical Information

CAS Number

2207-44-5
Formula Weight

295.36
Molecular Formula

C10H5N3O2S3
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 25 mg/mL (84.64 mM; Ultrasonic )
SMILES

O=[N+]([O-])C1=CN=C(SC2=NC3=C(S2)C=CC=C3)S1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Li P, et al. Discovery of a highly potent NPAS3 heterodimer inhibitor by covalently modifying ARNT. Bioorg Chem. 2023 Oct;139:106676.?

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