NESS-040C5

CAS No. 1445751-90-5

NESS-040C5( NESS 040C5 | NESS040C5 )

Catalog No. M11886 CAS No. 1445751-90-5

A potent, reasonably selective cannabinoid CB2 agonist with Ki of 0.4 nM, 25-fold selectivity over CB1 receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    NESS-040C5
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, reasonably selective cannabinoid CB2 agonist with Ki of 0.4 nM, 25-fold selectivity over CB1 receptor.
  • Description
    A potent, reasonably selective cannabinoid CB2 agonist with Ki of 0.4 nM, 25-fold selectivity over CB1 receptor.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    NESS 040C5 | NESS040C5
  • Pathway
    GPCR/G Protein
  • Target
    Cannabinoid Receptor
  • Recptor
    Cannabinoid Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1445751-90-5
  • Formula Weight
    447.64
  • Molecular Formula
    C27H33N3OS
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    ——
  • Chemical Name
    Thieno[3',2':4,5]cyclopenta[1,2-c]pyrazole-3-carboxamide, 1,4-dihydro-N-[5-methyl-2-(1-methylethyl)cyclohexyl]-1-[(4-methylphenyl)methyl]-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Hanus LO, et al. Curr Med Chem. 2010;17(14):1341-59.
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