MS0124

CAS No. 1197196-63-6

MS0124 ( MS 0124 )

Catalog No. M10701 CAS No. 1197196-63-6

MS-0124 is a potent and selective inhibitor of G9a-like Protein (GLP) lysine methyltransferase with IC50 of 13 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 718 Get Quote
10MG 981 Get Quote
25MG 1485 Get Quote
50MG 2007 Get Quote
100MG 2637 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    MS0124
  • Note
    Research use only, not for human use.
  • Brief Description
    MS-0124 is a potent and selective inhibitor of G9a-like Protein (GLP) lysine methyltransferase with IC50 of 13 nM.
  • Description
    MS-0124 is a potent and selective inhibitor of G9a-like Protein (GLP) lysine methyltransferase with IC50 of 13 nM, shows >30-fold selectivity for GLP over G9a and other methyltransferases.
  • Synonyms
    MS 0124
  • Pathway
    Chromatin/Epigenetic
  • Target
    HMTase
  • Recptor
    HMTase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1197196-63-6
  • Formula Weight
    387.48
  • Molecular Formula
    C20H29N5O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    COC1=CC2=NC(N3CCOCC3)=NC(NC4CCN(C)CC4)=C2C=C1OC
  • Chemical Name
    6,7-Dimethoxy-N-(1-methylpiperidin-4-yl)-2-morpholinoquinazolin-4-amine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Xiong Y, et al. J Med Chem. 2017 Mar 9;60(5):1876-1891.
molnova catalog
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