MS0124

CAS No. 1197196-63-6

MS0124( MS 0124 )

Catalog No. M10701 CAS No. 1197196-63-6

MS-0124 is a potent and selective inhibitor of G9a-like Protein (GLP) lysine methyltransferase with IC50 of 13 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 123 In Stock
5MG 117 In Stock
10MG 196 In Stock
25MG 392 In Stock
50MG 616 In Stock
100MG 861 In Stock
200MG 1144 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    MS0124
  • Note
    Research use only, not for human use.
  • Brief Description
    MS-0124 is a potent and selective inhibitor of G9a-like Protein (GLP) lysine methyltransferase with IC50 of 13 nM.
  • Description
    MS-0124 is a potent and selective inhibitor of G9a-like Protein (GLP) lysine methyltransferase with IC50 of 13 nM, shows >30-fold selectivity for GLP over G9a and other methyltransferases.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    MS 0124
  • Pathway
    Chromatin/Epigenetic
  • Target
    HMTase
  • Recptor
    HMTase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1197196-63-6
  • Formula Weight
    387.484
  • Molecular Formula
    C20H29N5O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    COC1=CC2=NC(N3CCOCC3)=NC(NC4CCN(C)CC4)=C2C=C1OC
  • Chemical Name
    6,7-Dimethoxy-N-(1-methylpiperidin-4-yl)-2-morpholinoquinazolin-4-amine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Xiong Y, et al. J Med Chem. 2017 Mar 9;60(5):1876-1891.
molnova catalog
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