MS0124

CAS No. 1197196-63-6

MS0124 ( MS 0124 )

Catalog No. M10701 CAS No. 1197196-63-6

MS-0124 is a potent and selective inhibitor of G9a-like Protein (GLP) lysine methyltransferase with IC50 of 13 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 718 Get Quote
10MG 981 Get Quote
25MG 1485 Get Quote
50MG 2007 Get Quote
100MG 2637 Get Quote
200MG Get Quote Get Quote
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Biological Information

  • Product Name
    MS0124
  • Note
    Research use only, not for human use.
  • Brief Description
    MS-0124 is a potent and selective inhibitor of G9a-like Protein (GLP) lysine methyltransferase with IC50 of 13 nM.
  • Description
    MS-0124 is a potent and selective inhibitor of G9a-like Protein (GLP) lysine methyltransferase with IC50 of 13 nM, shows >30-fold selectivity for GLP over G9a and other methyltransferases.
  • Synonyms
    MS 0124
  • Pathway
    Chromatin/Epigenetic
  • Target
    HMTase
  • Recptor
    HMTase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1197196-63-6
  • Formula Weight
    387.48
  • Molecular Formula
    C20H29N5O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    COC1=CC2=NC(N3CCOCC3)=NC(NC4CCN(C)CC4)=C2C=C1OC
  • Chemical Name
    6,7-Dimethoxy-N-(1-methylpiperidin-4-yl)-2-morpholinoquinazolin-4-amine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Xiong Y, et al. J Med Chem. 2017 Mar 9;60(5):1876-1891.
molnova catalog
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