MPEP

CAS No. 96206-92-7

MPEP ( —— )

Catalog No. M19286 CAS No. 96206-92-7

MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable activity at mGlu1b/2/3/4a/7b/8a/6 receptors.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
10MG 42 Get Quote
25MG 88 Get Quote
50MG 162 Get Quote
100MG 260 Get Quote
200MG 428 Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    MPEP
  • Note
    Research use only, not for human use.
  • Brief Description
    MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable activity at mGlu1b/2/3/4a/7b/8a/6 receptors.
  • Description
    MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable activity at mGlu1b/2/3/4a/7b/8a/6 receptors.
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    mGluR5
  • Research Area
    Neurological Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    96206-92-7
  • Formula Weight
    193.24
  • Molecular Formula
    C14H11N
  • Purity
    98%
  • Solubility
    ——
  • SMILES
    CC1=NC(=CC=C1)C#CC1=CC=CC=C1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Gasparini F, et al. Neuropharmacology, 1999, 38(10), 1493-1503.
molnova catalog
related products
  • Methyl isoeugenol

    methyl isoeugenol (MIE) is a natural food flavour that constitutes 93.7% of an essential oil from Pimenta pseudocaryophyllus leaf. The leaf extracts of this species are used as a calming agent. As a ubiquitous food additive the application of MIE for treating mood disorders.

  • Eliglustat hemitartr...

    Eliglustat Hemitartrate, with an IC50 of 24 nM, is a specific, potent, oral active glucocerebral glycosidase inhibitor.Eliglustat tartrate shows good potency with an IC50 of 24 nM and specificity against the target enzyme.A novel inhibitor of glucosylceramide synthase (Genz-112638) and assessed its activity in a murine model of Gaucher disease (D409V/null).?Biochemical characterization of Genz-112638 showed good potency (IC(50) approximately 24nM) and specificity against the target enzyme.?

  • SHMT-IN-1

    SHMT-IN-1 is a potent plasmodial serine hydroxymethyltransferase (SHMT) inhibitor,and with antitumor activity.