ML298

CAS No. 1426916-02-0

ML298( CID53393915 )

Catalog No. M23583 CAS No. 1426916-02-0

ML298 is a potent, specific inhibitor of Phospholipase D2 (PLD2, IC50 of 355 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 72 In Stock
10MG 115 In Stock
25MG 197 In Stock
50MG 293 In Stock
100MG 437 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
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Biological Information

  • Product Name
    ML298
  • Note
    Research use only, not for human use.
  • Brief Description
    ML298 is a potent, specific inhibitor of Phospholipase D2 (PLD2, IC50 of 355 nM).
  • Description
    ML298 is a potent, specific inhibitor of Phospholipase D2 (PLD2, IC50 of 355 nM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    CID53393915
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Phospholipase
  • Recptor
    PLD2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1426916-02-0
  • Formula Weight
    432.4
  • Molecular Formula
    C22H23F3N4O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:10 mM
  • SMILES
    C1CN(CCC12C(=O)NCN2C3=CC(=CC=C3)F)CCNC(=O)C4=CC(=C(C=C4)F)F
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Brown K A . Development of dual PLD1/2 and PLD2 selective inhibitors from a common 1,3,8-Triazaspiro[4.5]decane Core: discovery of Ml298 and Ml299 that decrease invasive migration in U87-MG glioblastoma cells.[J]. Journal of Medicinal Chemistry, 2013, 56(6):2695.
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