MK-2295
CAS No. 878811-00-8
MK-2295 ( MK2295; MK 2295 )
Catalog No. M27996 CAS No. 878811-00-8
MK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 393 | Get Quote |
|
10MG | 581 | Get Quote |
|
25MG | 888 | Get Quote |
|
50MG | 1242 | Get Quote |
|
100MG | 1674 | Get Quote |
|
500MG | 3348 | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameMK-2295
-
NoteResearch use only, not for human use.
-
Brief DescriptionMK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.
-
DescriptionMK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.
-
SynonymsMK2295; MK 2295
-
PathwayMembrane Transporter/Ion Channel
-
TargetTRP/TRPV Channel
-
RecptorJAK1
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number878811-00-8
-
Formula Weight490.6
-
Molecular FormulaC27H31FN6O2
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESC[C@@H]1CCCN1c1nc(cc(n1)-c1ccc(F)cc1)N1CCN(C[C@H]1C)c1ncc(cc1C)C(O)=O
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Paul Smith, et al. Use of jak1 inhibitors for the treatment of cutaneous lupus erythematosus and lichen planus (lp). WO2021076124A1.
molnova catalog
related products
-
AMG-9810
A potent, selective and competitive TRPV1 antagonist with IC50 of 24.5 and 85.6 nM for human and rat TRPV1, repectively.
-
Capsaicin
Capsaicin is an active component of chili peppers. It selectively binds to TRPV1 which is a heat-activated calcium channel.
-
JNJ-38893777 sulfate
JNJ-38893777 is a potent and selective transient receptor potential vanilloid 1 (TRPV1) channel antagonist for treatment of ociceptive and neuropathic pain.