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MK-2295
CAS No. 878811-00-8
MK-2295( MK2295 | MK 2295 )
Catalog No. M27996 CAS No. 878811-00-8
MK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 393 | Get Quote |
|
| 10MG | 581 | Get Quote |
|
| 25MG | 888 | Get Quote |
|
| 50MG | 1242 | Get Quote |
|
| 100MG | 1674 | Get Quote |
|
| 500MG | 3348 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameMK-2295
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NoteResearch use only, not for human use.
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Brief DescriptionMK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.
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DescriptionMK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.
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In Vitro——
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In Vivo——
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SynonymsMK2295 | MK 2295
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PathwayMembrane Transporter/Ion Channel
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TargetTRP/TRPV Channel
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RecptorJAK1
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Research Area——
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Indication——
Chemical Information
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CAS Number878811-00-8
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Formula Weight490.583
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Molecular FormulaC27H31FN6O2
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Purity>98% (HPLC)
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Solubility——
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SMILESC[C@@H]1CCCN1c1nc(cc(n1)-c1ccc(F)cc1)N1CCN(C[C@H]1C)c1ncc(cc1C)C(O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Paul Smith, et al. Use of jak1 inhibitors for the treatment of cutaneous lupus erythematosus and lichen planus (lp). WO2021076124A1.
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