
MB-07811
CAS No. 852948-13-1
MB-07811( VK-2809 )
Catalog No. M26750 CAS No. 852948-13-1
MB-07811 is an orally active HepDirect prodrug of MB07344 with cholesterol and triglycerides lowering activity. MB-07811 is an agonist of liver-targeted THR-β.
Purity : >98% (HPLC)






Size | Price / USD | Stock | Quantity |
5MG | 393 | Get Quote |
![]() ![]() |
10MG | 581 | Get Quote |
![]() ![]() |
25MG | 888 | Get Quote |
![]() ![]() |
50MG | 1242 | Get Quote |
![]() ![]() |
100MG | Get Quote | Get Quote |
![]() ![]() |
200MG | Get Quote | Get Quote |
![]() ![]() |
500MG | Get Quote | Get Quote |
![]() ![]() |
1G | Get Quote | Get Quote |
![]() ![]() |
Biological Information
-
Product NameMB-07811
-
NoteResearch use only, not for human use.
-
Brief DescriptionMB-07811 is an orally active HepDirect prodrug of MB07344 with cholesterol and triglycerides lowering activity. MB-07811 is an agonist of liver-targeted THR-β.
-
DescriptionMB-07811 is an orally active HepDirect prodrug of MB07344 with cholesterol and triglycerides lowering activity. MB-07811 is an agonist of liver-targeted THR-β.(In Vitro):MB-07811 has a low affinity for thyroid hormone receptors with a Ki of 14.6 μM for TRβ and a Ki of 12.5 μM for TRα.(In Vivo):In diet-induced obese mice, MB-07811 (0.3-30 mg/kg) decreases cholesterol and triglycerides.
-
In Vitro——
-
In Vivo——
-
SynonymsVK-2809
-
PathwayEndocrinology/Hormones
-
TargetTHR
-
RecptorSST2
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number852948-13-1
-
Formula Weight514.98
-
Molecular FormulaC28H32ClO5P
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESCC(C)c1cc(Cc2c(C)cc(OC[P@@]3(=O)OCC[C@H](O3)c3cccc(Cl)c3)cc2C)ccc1O
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Murray B. Gordon, et al. Identification of a dose range for once daily oral paltusotine in patients with acromegaly that maintains IGF-1 levels when switching from long-acting somatostatin receptor ligand therapy. Endocrine Abstracts (2021) 73 OC15.4.
molnova catalog



related products
-
TR antagonist 1
TR antagonist 1 is a highly potent thyroid hormone receptor (TR) antagonist (IC50 of 36 and 22 nM for TRα and TRβ, respectively) that can be used to study diseases caused by endocrine abnormalities.
-
Triiodothyronine Sul...
Triiodothyronine Sulfate is a prodrug to the Conventional Hormone Therapy of Hypothyroidism.
-
Parathyroid Hormone ...
Parathyroid Hormone (1-34), bovine, a parathyroid hormone (PTH) receptor agonist from the parathyroid hormone family, is used to study osteoporosis and hypoparathyroidism.