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Antide
CAS No. 112568-12-4
Antide( ——— )
Catalog No. M40004 CAS No. 112568-12-4
Antide (D-21074) is a potent LHRH antagonist. Antide also can be used for the research of prostatic cancer.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 171 | In Stock |
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| 10MG | 283 | In Stock |
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| 25MG | Get Quote | In Stock |
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| 50MG | Get Quote | In Stock |
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| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameAntide
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NoteResearch use only, not for human use.
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Brief DescriptionAntide (D-21074) is a potent LHRH antagonist. Antide also can be used for the research of prostatic cancer.
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DescriptionAntide (D-21074) is a potent LHRH antagonist. Antide also can be used for the research of prostatic cancer.
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In Vitro———
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In VivoAnimal Model:Cynomolgus monkey and rat Dosage:1, 3, 6, 10 and 15 mg/kg Administration:Subcutaneous, once or on 5 consecutive days Result:Had a dose-dependent inhibitory effect on serum concentration of LH (only rat) and testosterone and on the weights of the testes, prostates and seminal vesicles.Achieved long-lasting castration-like effects at concentrations between 6 (less than or equal to 8 weeks) and 15 mg/kg (greater than 8 weeks) in the rat. Induced a prolonged inhibitory effect only at 15 mg/kg and the duration was only 2-3 weeks in the cynomolgus monkey.
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Synonyms———
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PathwayOthers
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TargetOther Targets
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Recptor———
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Research Area———
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Indication———
Chemical Information
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CAS Number112568-12-4
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Formula Weight1591.29
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Molecular FormulaC82H108ClN17O14
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Purity>98% (HPLC)
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SolubilityH2O : 10 mg/mL (6.28 mM; ultraphonic)
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SMILES———
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. U F Habenicht, et al. Effect of the new potent LHRH antagonist antide. J Steroid Biochem Mol Biol. 1990 Dec 20;37(6):937-42. ?
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