C 101248

CAS No. 361368-24-3

C 101248( —— )

Catalog No. M37356 CAS No. 361368-24-3

C 101248 is a selective and potent inhibitor targeting both mouse and human tandem pore domain halothane-inhibited K+ channel 1 (THIK-1, IC50= 50 nM), without affecting the K2P family members (TREK-1, TWIK-2) and Kv2.1.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 188 In Stock
10MG 282 In Stock
25MG 489 In Stock
50MG 695 In Stock
100MG 977 In Stock
200MG Get Quote In Stock
500MG 1934 In Stock
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Biological Information

  • Product Name
    C 101248
  • Note
    Research use only, not for human use.
  • Brief Description
    C 101248 is a selective and potent inhibitor targeting both mouse and human tandem pore domain halothane-inhibited K+ channel 1 (THIK-1, IC50= 50 nM), without affecting the K2P family members (TREK-1, TWIK-2) and Kv2.1.
  • Description
    KCNK13-IN-1 (example 71), a KCNK13 antagonist, is an anti-inflammatory agent, with an IC50 of <200 nM for IL-1 β.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    Others
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    361368-24-3
  • Formula Weight
    292.3
  • Molecular Formula
    C15H12N6O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    NC1=NON=C1C2=NC3=CC=CC=C3N2CC4=CC=NC=C4
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Roland BüRLI, et al. Novel compounds. Patent WO2022167819.
molnova catalog
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