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AChE/BuChE-IN-4
CAS No. 1997158-25-4
AChE/BuChE-IN-4( —— )
Catalog No. M37106 CAS No. 1997158-25-4
AChE/BuChE-IN-4 is a multi-target AChE/BuChE inhibitor with oral activity and blood-brain barrier permeability, with IC50 values of 2.08 and 7.41 μM for AChE and BuChE, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 105 | In Stock |
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| 10MG | 159 | In Stock |
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| 25MG | 235 | In Stock |
|
| 50MG | 310 | In Stock |
|
| 100MG | 461 | In Stock |
|
| 200MG | 624 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameAChE/BuChE-IN-4
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NoteResearch use only, not for human use.
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Brief DescriptionAChE/BuChE-IN-4 is a multi-target AChE/BuChE inhibitor with oral activity and blood-brain barrier permeability, with IC50 values of 2.08 and 7.41 μM for AChE and BuChE, respectively.
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DescriptionAChE/BuChE-IN-4(compound 4a) is aorally activeandbrain-penetrantmultitarget-directedAChE/BuChEinhibitor againstAChEandBuChE, with theIC50of 2.08 and 7.41 μM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetAChE
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RecptorAChE
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Research Area——
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Indication——
Chemical Information
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CAS Number1997158-25-4
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Formula Weight297.4
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Molecular FormulaC17H23N5
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Purity>98% (HPLC)
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Solubility——
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SMILESN=1C=CC(=NC1N)NCC2CCN(CC=3C=CC=CC3)CC2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Concei??o RAD, et al. Structure-based design of new N-benzyl-piperidine derivatives as multitarget-directed AChE/BuChE inhibitors for Alzheimer's disease [published online ahead of print, 2023 Oct 5]. J Cell Biochem. 2023;10.1002/jcb.30483.?
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