Cart
sales@molnova.com
ERK5-IN-6
CAS No. 2734916-64-2
ERK5-IN-6( —— )
Catalog No. M37089 CAS No. 2734916-64-2
ERK5-IN-6 is a potent inhibitor of ERK5 kinase.ERK5-IN-6 exhibits antiproliferative activity, anticonvulsant activity, and antitumor activity, and can be used in the study of central nervous system-related disorders.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 296 | In Stock |
|
| 5MG | 459 | In Stock |
|
| 10MG | 657 | In Stock |
|
| 25MG | 994 | In Stock |
|
| 50MG | 1371 | In Stock |
|
| 100MG | 1773 | In Stock |
|
| 500MG | 3537 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameERK5-IN-6
-
NoteResearch use only, not for human use.
-
Brief DescriptionERK5-IN-6 is a potent inhibitor of ERK5 kinase.ERK5-IN-6 exhibits antiproliferative activity, anticonvulsant activity, and antitumor activity, and can be used in the study of central nervous system-related disorders.
-
DescriptionERK5-IN-6 (compound 5J)is an ERK5 kinase inhibitor with anticancer activity. ERK5-IN-6 exhibits good anti-proliferative activity with the IC50 value of 4.56 μg/mL for A549 cells.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayMAPK/ERK Signaling
-
TargetERK
-
RecptorERK
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number2734916-64-2
-
Formula Weight339.43
-
Molecular FormulaC23H21N3
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESN1=CC=CC2=C1NC=C2C3=CCN(CC=4C=CC=5C=CC=CC5C4)CC3
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Qin Zhang, et al. Design, synthesis and SAR of novel 7-azaindole derivatives as potential Erk5 kinase inhibitor with anticancer activity. Bioorg Med Chem. 2023 Oct 14:95:117503. ?
molnova catalog
related products
-
DEL-22379
A small molecule inhibitor of ERK dimerization with IC50 of 0.5 uM, without affecting ERK phosphorylation.
-
ERK-IN-3
ERK-IN-3 is a potent and orally active inhibitor of ERK. It inhibits ERK1/2 with low single-digit nM IC50 values. It can be used for the research of cancers driven by RAS mutations.
-
MK-8353
MK-8353 (SCH-900353) is a?highly potent, orally bioavailable, dual-specificity ERK1/2 inhibitor with IC50 of 23.0/8.8 nM, respectively.
