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Nav1.8-IN-4
CAS No. 1620846-16-3
Nav1.8-IN-4( —— )
Catalog No. M37057 CAS No. 1620846-16-3
Nav1.8-IN-4 is a potent Nav1.8 channel inhibitor with potential analgesic activity.Nav1.8-IN-4 can be used for pain and neurological related disorders.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 73 | In Stock |
|
| 5MG | 121 | In Stock |
|
| 10MG | 188 | In Stock |
|
| 25MG | 376 | In Stock |
|
| 50MG | 600 | In Stock |
|
| 100MG | 918 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | 1841 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameNav1.8-IN-4
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NoteResearch use only, not for human use.
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Brief DescriptionNav1.8-IN-4 is a potent Nav1.8 channel inhibitor with potential analgesic activity.Nav1.8-IN-4 can be used for pain and neurological related disorders.
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DescriptionNav1.8-IN-4 (compound 9a) is a Nav1.8 channel inhibitor (IC50=0.014 μM). Nav1.8-IN-4 can be used for research on pain-related diseases.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetSodium Channel
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RecptorSodium Channel
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Research Area——
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Indication——
Chemical Information
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CAS Number1620846-16-3
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Formula Weight406.33
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Molecular FormulaC20H14F4N2O3
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (307.63 mM; Ultrasonic )
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SMILESO=C1C=C(C=CN1)NC(=O)C2=CC=C(C=C2OC3=CC=C(F)C=C3C)C(F)(F)F
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Corey Anderson, et al. Prodrugs of pyridone amides useful as modulators of sodium channels. Patent WO2015089361A1.
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