hTYR/AbTYR-IN-1

CAS No. 1625821-37-5

hTYR/AbTYR-IN-1( —— )

Catalog No. M37018 CAS No. 1625821-37-5

hTYR/AbTYR-IN-1 is a dual hTYR/AbTYR inhibitor with inhibitory effects on hTYR and AbTYR, with IC50s of 5.4 μM and 3.52 μM, respectively.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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25MG 70 In Stock
50MG 101 In Stock
100MG 151 In Stock
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Biological Information

  • Product Name
    hTYR/AbTYR-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    hTYR/AbTYR-IN-1 is a dual hTYR/AbTYR inhibitor with inhibitory effects on hTYR and AbTYR, with IC50s of 5.4 μM and 3.52 μM, respectively.
  • Description
    hTYR/AbTYR-IN-1 (Compound 7) is a hTYR/AbTYR dual inhibitor, with IC50s of 5.4 μM and 3.52 μM for hTYR and AbTYR respectively.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Proteasome/Ubiquitin
  • Target
    Tyrosinase
  • Recptor
    Tyrosinase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1625821-37-5
  • Formula Weight
    312.36
  • Molecular Formula
    C18H20N2O3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 125 mg/mL (400.18 mM; Ultrasonic )
  • SMILES
    C(=O)(C1=C(OC)C=CC=C1)N2CCN(CC2)C3=CC=C(O)C=C3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Ricci F, et al. Computational methods to analyze and predict the binding mode of inhibitors targeting both human and mushroom tyrosinase. Eur J Med Chem. 2023 Aug 28;260:115771.?
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