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Zelasudil
CAS No. 2365193-22-0
Zelasudil( —— )
Catalog No. M36300 CAS No. 2365193-22-0
Zelasudil (RXC007) is a Rho-related (ROCK) kinase inhibitor for the study of idiopathic pulmonary fibrosis and inflammation.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 188 | In Stock |
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| 5MG | 180 | In Stock |
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| 10MG | 275 | In Stock |
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| 25MG | 468 | In Stock |
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| 50MG | 640 | In Stock |
|
| 100MG | 892 | In Stock |
|
| 200MG | 1200 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameZelasudil
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NoteResearch use only, not for human use.
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Brief DescriptionZelasudil (RXC007) is a Rho-related (ROCK) kinase inhibitor for the study of idiopathic pulmonary fibrosis and inflammation.
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DescriptionZelasudil is a Rho-associated (ROCK) kinase inhibitor. Zelasudil has a ROCK2 binding affinity.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetROCK
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RecptorROCK
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Research Area——
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Indication——
Chemical Information
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CAS Number2365193-22-0
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Formula Weight437.445
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Molecular FormulaC22H21F2N7O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (228.60 mM; Ultrasonic )
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SMILESO=C(NCC(F)F)C=1C=CC(=CC1)C=2N=C(NC3=CC=C4NN=CC4=C3C5CC5)N(N2)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Lee E, et al. Selective ROCK2 inhibition for treatment of edema and associated conditions: World Intellectual Property Organization, WO2022169946. 2022-08-11.
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