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GAC0003A4
CAS No. 929492-71-7
GAC0003A4( —— )
Catalog No. M36252 CAS No. 929492-71-7
GAC0003A4 is a potent LXR inverse agonist with antitumor activity that inhibits the transcription of LXR proteins.GAC0003A4 degrades LXRβ proteins and inhibits the proliferation of PDAC cells in a dose-dependent manner.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 159 | In Stock |
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| 10MG | 252 | In Stock |
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| 25MG | 418 | In Stock |
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| 50MG | 577 | In Stock |
|
| 100MG | 775 | In Stock |
|
| 200MG | 1042 | In Stock |
|
| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameGAC0003A4
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NoteResearch use only, not for human use.
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Brief DescriptionGAC0003A4 is a potent LXR inverse agonist with antitumor activity that inhibits the transcription of LXR proteins.GAC0003A4 degrades LXRβ proteins and inhibits the proliferation of PDAC cells in a dose-dependent manner.
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DescriptionGAC0003A4 is an LXR inverse agonist that inhibits LXR transcriptional activity. GAC0003A4 also efficiently degrades LXRβ protein. GAC0003A4 has the potential to be used in advanced pancreatic cancer and other refractory malignancies.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorLiver X Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number929492-71-7
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Formula Weight340.42
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Molecular FormulaC20H24N2O3
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (367.19 mM; Ultrasonic )
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SMILESC(=O)(C1=CC(OC)=CC(OC)=C1)N2CCN(CC2)C3=C(C)C=CC=C3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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