Saterinone
CAS No. 102669-89-6
Saterinone( —— )
Catalog No. M36223 CAS No. 102669-89-6
Saterinone is a potent and selective phosphodiesterase III inhibitor and a potent antagonist of the vascular α-1-adrenoceptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 183 | In Stock |
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| 5MG | 155 | In Stock |
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| 10MG | 235 | In Stock |
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| 25MG | 376 | In Stock |
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| 50MG | 500 | In Stock |
|
| 100MG | 671 | In Stock |
|
| 200MG | 905 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSaterinone
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NoteResearch use only, not for human use.
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Brief DescriptionSaterinone is a potent and selective phosphodiesterase III inhibitor and a potent antagonist of the vascular α-1-adrenoceptor.
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DescriptionSaterinone is a potent and selective phosphodiesterase III inhibitor and a potent antagonist of the vascular α-1-adrenoceptor. Saterinone has vasodilatory properties and can be used in the acute treatment of chronic heart failure. Saterinone inhibited crude cAMP phosphodiesterase (PDE) activity in guinea pig right ventricular homogenates The ic50 value is 2.3 × 10(-5) mol/l.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetAdrenergic Receptor
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RecptorAdrenergic Receptor | PDE
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Research Area——
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Indication——
Chemical Information
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CAS Number102669-89-6
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Formula Weight474.55
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Molecular FormulaC27H30N4O4
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Purity>98% (HPLC)
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Solubility——
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SMILESCC1=C(C=C(C#N)C(=O)N1)C2=CC=C(OCC(CN3CCN(CC3)C4=C(OC)C=CC=C4)O)C=C2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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