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HDAC-IN-52
CAS No. 2075787-77-6
HDAC-IN-52( —— )
Catalog No. M36045 CAS No. 2075787-77-6
HDAC-IN-52, a pyridine-containing HDAC inhibitor, effectively inhibits HDAC1, HDAC2, HDAC3, and HDAC10 with IC50 values of 0.189, 0.227, 0.440, and 0.446 μM, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 179 | In Stock |
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| 5MG | 157 | In Stock |
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| 10MG | 234 | In Stock |
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| 25MG | 356 | In Stock |
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| 50MG | 476 | In Stock |
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| 100MG | 644 | In Stock |
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| 200MG | 866 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameHDAC-IN-52
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NoteResearch use only, not for human use.
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Brief DescriptionHDAC-IN-52, a pyridine-containing HDAC inhibitor, effectively inhibits HDAC1, HDAC2, HDAC3, and HDAC10 with IC50 values of 0.189, 0.227, 0.440, and 0.446 μM, respectively.
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DescriptionHDAC-IN-52 is a pyridine-containing HDAC inhibitor, with IC50s of 0.189, 0.227, 0.440 and 0.446 μM for HDAC1, HDAC2, HDAC3, and HDAC10, respectively. HDAC-IN-52 can be used for the research of cancer.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetHDAC
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RecptorHDAC
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Research Area——
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Indication——
Chemical Information
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CAS Number2075787-77-6
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Formula Weight396.44
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Molecular FormulaC24H20N4O2
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Purity>98% (HPLC)
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Solubility——
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SMILESC(C(NC=1C=CC(C(NC2=C(N)C=CC=C2)=O)=NC1)=O)C3=CC4=C(C=C3)C=CC=C4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Bello ED, et, al. Novel pyridine-containing histone deacetylase inhibitors strongly arrest proliferation, induce apoptosis and modulate miRNAs in cancer cells. Eur J Med Chem. 2022 Dec 15;247:115022.?
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