5-LOX-IN-1

CAS No. 55040-82-9

5-LOX-IN-1( —— )

Catalog No. M35529 CAS No. 55040-82-9

5-LOX-IN-1 is a 5-Lipoxygenase (5-LOX) inhibitor (IC50: 2.3 μM).5-LOX-IN-1 can be used for cancer research.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 45 Get Quote
10MG 76 Get Quote
25MG 150 Get Quote
50MG 227 Get Quote
100MG 335 Get Quote
500MG 782 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    5-LOX-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    5-LOX-IN-1 is a 5-Lipoxygenase (5-LOX) inhibitor (IC50: 2.3 μM).5-LOX-IN-1 can be used for cancer research.
  • Description
    5-LOX-IN-1 (compound 2b) is an inhibitor of human 5-Lipoxygenase (5-LOX) with an IC50 value of 2.3 μM. 5-LOX-IN-1 can be used for the research of inflammation.
  • In Vitro
    5-LOX-IN-1 (0-10 μM) inhibits 5-LOX with an IC50 value of 2.3 μM.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Immunology/Inflammation
  • Target
    Lipoxygenase
  • Recptor
    Lipoxygenase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    55040-82-9
  • Formula Weight
    350.43
  • Molecular Formula
    C20H18N2O2S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (285.36 mM; Ultrasonic (<60°C)
  • SMILES
    O=C(c1sc(nc1-c1ccccc1)N1CCOCC1)c1ccccc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Sinha S, et al. Design, synthesis and identification of novel substituted 2-amino thiazole analogues as potential anti-inflammatory agents targeting 5-lipoxygenase. Eur J Med Chem. 2018 Oct 5;158:34-50.?
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