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Legumain inhibitor 1
CAS No. 2361157-34-6
Legumain inhibitor 1( —— )
Catalog No. M35166 CAS No. 2361157-34-6
Legumain inhibitor 1 is a highly potent and specific Legumain inhibitor with potential anticancer activity for cancer research.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 454 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameLegumain inhibitor 1
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NoteResearch use only, not for human use.
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Brief DescriptionLegumain inhibitor 1 is a highly potent and specific Legumain inhibitor with potential anticancer activity for cancer research.
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DescriptionLegumain inhibitor 1 is a potent and selective Legumain inhibitor with an IC50 of 3.6 nM. Legumain inhibitor 1 can be used for cancer research.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayNeuroscience
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TargetGamma-secretase
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RecptorGamma-secretase
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Research Area——
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Indication——
Chemical Information
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CAS Number2361157-34-6
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Formula Weight467.54
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Molecular FormulaC23H25N5O4S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 40 mg/mL (85.55 mM; Ultrasonic )
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SMILESCn1ncc2cc(ccc12)-c1ccc(cc1)S(=O)(=O)CC(C)(C)C(=O)N[C@@H](CC(N)=O)C#N
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Sharon L Eddie, et al. Identification and SAR exploration of a novel series of Legumain inhibitors. Bioorg Med Chem Lett. 2019 Jun 15;29(12):1546-1548.?
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