Cart
sales@molnova.com
PKA-IN-1
CAS No. 179985-52-5
PKA-IN-1( —— )
Catalog No. M35100 CAS No. 179985-52-5
PKA-IN-1 is a selective and potent cyclic AMP-dependent protein kinase (PKA) catalytic subunit (cAK) inhibitor (IC50: 0.03 μM).PKA-IN-1 can be used to study diseases of the immune system.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 10MG | 37 | Get Quote |
|
| 25MG | 59 | Get Quote |
|
| 50MG | 90 | Get Quote |
|
| 100MG | 140 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NamePKA-IN-1
-
NoteResearch use only, not for human use.
-
Brief DescriptionPKA-IN-1 is a selective and potent cyclic AMP-dependent protein kinase (PKA) catalytic subunit (cAK) inhibitor (IC50: 0.03 μM).PKA-IN-1 can be used to study diseases of the immune system.
-
DescriptionPKA-IN-1 is a potent and selective cyclic AMP-dependent protein kinase (PKA) catalytic subunit (cAK) inhibitor with an IC50 of 0.03 μM.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayApoptosis
-
TargetPKA
-
RecptorPKA
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number179985-52-5
-
Formula Weight225.25
-
Molecular FormulaC13H11N3O
-
Purity>98% (HPLC)
-
SolubilityIn Vitro:?DMSO : 62.5 mg/mL (277.47 mM; Ultrasonic (<80°C)
-
SMILESCC(=O)Nc1nc(C)c(C#N)c2ccccc12
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Z X Lu, et al. Selective inhibition of cyclic AMP-dependent protein kinase by isoquinoline derivative. Biol Chem Hoppe Seyler. 1996 Jun;377(6):373-8?
molnova catalog
related products
-
Pomolic acid
Pomolic acid has anti-cancer, anti-inflammatory and apoptotic activities.
-
CREBtide
CREBtide is a synthetic substrate for PKA (Km=3.9 μM), which is based on the phosphorylation sequence in d-CREB (cAMP response element binding protein).
-
HA-100
HA-100 is an inhibitor of protein kinase.
